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BT
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(IO-202)Tj
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(+)Tj
0.75 0 Td
(Azacitidine)Tj
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(LILRB4)Tj
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(antibody)Tj
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(Updated February 2023)Tj
/T1_0 1 Tf
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0.655 0.663 0.675 rg
(\037)Tj
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( )Tj
(2: Acquired by Morphosys )Tj
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(\037)Tj
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( )Tj
(3: Licensed from University of Michigan)Tj
/T1_2 1 Tf
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(Magrolimab)Tj
0 -1.2 Td
(+ Azacitidine)Tj
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(CD47)Tj
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(antibody)Tj
ET
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f
Q
0.773 0.412 0.373 rg
q 1 0 0 1 1942.8184 1427.9769 cm
0 0 m
-0.532 0.231 -0.623 0.726 -0.729 1.213 c
-0.486 0.809 -0.243 0.404 0 0 c
f
Q
q 1 0 0 1 1939.1946 1432.1189 cm
0 0 m
-0.378 -0.062 -0.619 0.101 -0.746 0.452 c
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f
Q
q 1 0 0 1 1939.912 1431.6217 cm
0 0 m
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h
f
Q
q 1 0 0 1 1940.1709 1431.3949 cm
0 0 m
-0.087 0.076 -0.175 0.152 -0.262 0.229 c
-0.175 0.153 -0.087 0.076 0 0 c
f
Q
q 1 0 0 1 1942.09 1429.1902 cm
0 0 m
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-0.089 0.132 -0.045 0.066 0 0 c
f
Q
Q
BT
24 0 0 24 2107.5137 1429.0449 Tm
(1)Tj
ET
q
1196.518 1124.116 387.69 132.999 re
W n
q
387.6904786 0 0 133.0000008 1196.517334 1124.115966 cm
/Im2 Do
Q
Q
BT
24 0 0 24 672.1479 844.8633 Tm
(Smoldering)Tj
0 -1.2 Td
(myeloma)Tj
0.008 7.961 Td
(AML/MDS)Tj
-0.043 4.843 Td
(NHL/MM)Tj
0.049 2.594 Td
(AML/CMML)Tj
0.064 9.528 Td
(MDS)Tj
-24.605 -14.6 Td
(ICT01)Tj
11.902 0.678 Td
[(B)14 (TN3A)]TJ
0 -1.2 Td
(antibody)Tj
12.579 0.461 Td
(heme malignancies)Tj
ET
q
1298.099 1040.283 179.302 59.999 re
W n
q
179.3023192 0 0 59.9999979 1298.0992432 1040.2825949 cm
/Im3 Do
Q
Q
q
0 1866.667 2505.333 -1866.667 re
W n
0.667 0 0 rg
0.667 0 0 RG
2419.75 1454.128 -2347.311 75.705 re
B
Q
BT
1 1 1 rg
27 0 0 27 2216.6855 1500.8076 Tm
[(R)30 (egulatory)]TJ
-0.509 -1.2 Td
(Designations)Tj
ET
q
0 1866.667 2505.333 -1866.667 re
W n
0.8 0.125 0.153 rg
2218 1405.333 -60 40 re
f
Q
BT
0 0 0 rg
24 0 0 24 86.3013 1256.959 Tm
(AFM13)Tj
0 -1.2 Td
(+)Tj
0.75 0 Td
[(NK)50 (-cells)]TJ
11.033 1.27 Td
[(CD30/CD16)6.9 (A)]TJ
0 -1.2 Td
(bispeci\037c engager)Tj
12.63 0.614 Td
(CD30+ lymphoma)Tj
ET
q
1536.999 1230.333 290.966 45 re
W n
q
290.9659029 0 0 44.999999 1536.9997559 1230.333497 cm
/Im4 Do
Q
Q
q
0 1866.667 2505.333 -1866.667 re
W n
0.8 0.125 0.153 rg
2218 1230.333 -60 40 re
f
0.659 0.667 0.675 rg
2311 1406.333 -60 40 re
f
Q
BT
24 0 0 24 84.9805 1374.6338 Tm
[(P)17 (elabresib)]TJ
0 -1.2 Td
[(+ Rux)24 (olitinib)]TJ
11.88 1.181 Td
(BET)Tj
0 -1.2 Td
(small molecule)Tj
ET
q
192.5925863 0 0 99.9999967 1882.2503662 1314.4139437 cm
/Im5 Do
Q
BT
24 0 0 24 2070.9404 1368.0352 Tm
(2)Tj
-58.276 -0.275 Td
(MPN)Tj
ET
q
0 1866.667 2505.333 -1866.667 re
W n
0.8 0.125 0.153 rg
2218 1347.333 -60 40 re
f
0.659 0.667 0.675 rg
2311 1347.333 -60 40 re
f
0 0 0 rg
2403 1406.333 -60 40 re
f
Q
BT
1 1 1 rg
27 0 0 27 83.7354 1482.8076 Tm
(Therapy)Tj
10.474 0 Td
[(T)78 (arget/Modality)]TJ
24.889 -0.024 Td
(Preclinical)Tj
19.978 0.493 Td
(Phase 1 Expand/)Tj
1.888 -1.2 Td
(Phase 2)Tj
-10.599 0.731 Td
(Phase 1)Tj
20.766 0.481 Td
[(Phase 2 R)30.1 (eg/)]TJ
1.175 -1.2 Td
(Phase 3)Tj
-46.769 0.706 Td
(Indications)Tj
0 0 0 rg
24 0 0 24 86.4277 1299.499 Tm
(Ziftomenib)Tj
11.799 0.677 Td
(Menin)Tj
0 -1.2 Td
(small molecule)Tj
ET
q
1855 1272.334 242.857 69.999 re
W n
q
242.8571486 0 0 70.0000017 1855 1272.3333724 cm
/Im6 Do
Q
Q
BT
24 0 0 24 2082.7617 1320.0811 Tm
(3)Tj
-58.827 -0.774 Td
(NPM1 mutant AML)Tj
ET
q
0 1866.667 2505.333 -1866.667 re
W n
0.8 0.125 0.153 rg
2218 1290.333 -60 40 re
f
2218 1111.333 -60 40 re
f
2218 994.333 -60 40 re
f
2218 1171.333 -60 40 re
f
2218 819.407 -60 40 re
f
0.659 0.667 0.675 rg
2311 1171.333 -60 40 re
f
0.8 0.125 0.153 rg
2218 701.333 -60 40 re
f
0.871 0.875 0.882 rg
2420.239 222.015 -2347.811 58.637 re
B
Q
BT
24 0 0 24 85.3242 711.4971 Tm
[(KT)60 (-333)]TJ
11.953 -0.019 Td
[(S)7 (T)64 (A)64 (T)7 (3 degrader)]TJ
-12.01 2.523 Td
[(B)14 (TX)47 (-1188)]TJ
11.923 0.667 Td
(GSPT1 + IKZF1/3 )Tj
0 -1.2 Td
(degrader)Tj
ET
q
0 1866.667 2505.333 -1866.667 re
W n
0.996 0.996 0.996 rg
q 1 0 0 1 1261.7412 694.1592 cm
0 0 m
-0.004 0 l
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4.635 -2.105 5.616 2.016 6.562 6.145 c
6.777 7.079 6.35 7.517 5.397 7.506 c
4.133 7.491 2.869 7.512 1.606 7.506 c
0.472 7.5 -0.065 7.002 -0.019 5.786 c
0.053 3.86 0 1.929 0 0 c
0.1 52.05 m
0.1 47.415 0.077 43.089 0.134 38.764 c
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2.677 37.239 4.52 37.068 6.656 37.607 c
5.452 42.594 4.296 47.382 3.117 52.268 c
1.96 52.184 1.127 52.124 0.1 52.05 c
65.924 5.705 m
66.815 5.662 67.402 5.607 67.99 5.611 c
69.854 5.624 69.934 5.689 69.948 7.49 c
69.968 9.954 69.87 12.423 69.989 14.881 c
70.048 16.112 70.224 17.456 70.78 18.523 c
72.431 21.691 74.073 24.908 76.141 27.804 c
78.292 30.819 79.862 34.111 81.609 37.326 c
81.809 37.694 81.853 38.148 81.973 38.573 c
78.74 39.236 78.305 39.136 76.719 36.614 c
75.16 34.135 73.761 31.556 72.286 29.024 c
71.794 28.179 71.083 27.403 70.824 26.494 c
70.332 24.766 69.431 23.418 68.028 22.348 c
66.905 22.771 66.442 23.653 65.927 24.584 c
63.555 28.871 61.13 33.13 58.682 37.374 c
57.687 39.097 55.269 39.4 53.646 38.123 c
55 35.577 56.335 33.032 57.704 30.506 c
58.236 29.525 58.844 28.585 59.42 27.629 c
61.293 24.518 63.246 21.452 64.997 18.274 c
65.575 17.226 65.832 15.898 65.884 14.684 c
66.009 11.768 65.924 8.844 65.924 5.705 c
151.203 20.71 m
152.266 20.763 153.05 20.832 153.834 20.835 c
157.902 20.85 161.97 20.827 166.038 20.864 c
167.539 20.877 168.138 21.673 167.862 22.999 c
167.645 24.045 166.927 24.118 166.064 24.115 c
161.863 24.096 157.661 24.096 153.46 24.111 c
151.501 24.118 151.223 24.393 151.207 26.267 c
151.188 28.601 151.18 30.935 151.195 33.269 c
151.21 35.555 151.309 35.647 153.566 35.648 c
158.167 35.65 162.769 35.625 167.37 35.645 c
169.039 35.652 169.583 36.364 169.205 37.867 c
168.903 39.064 167.927 38.848 167.099 38.851 c
161.231 38.87 155.362 38.873 149.494 38.865 c
147.336 38.862 147.258 38.768 147.256 36.583 c
147.248 26.98 147.241 17.377 147.244 7.774 c
147.244 7.132 147.327 6.489 147.368 5.901 c
147.739 5.771 147.923 5.652 148.107 5.651 c
154.708 5.629 161.31 5.624 167.911 5.599 c
168.987 5.595 169.257 6.168 169.257 7.123 c
169.256 8.126 169.034 8.844 167.845 8.823 c
167.245 8.812 166.645 8.831 166.045 8.831 c
161.777 8.832 157.509 8.817 153.241 8.839 c
151.819 8.846 151.24 9.269 151.221 10.454 c
151.168 13.781 151.203 17.11 151.203 20.71 c
14.297 38.852 m
14.297 37.887 14.297 37.17 14.297 36.453 c
14.295 29.32 14.292 22.186 14.293 15.053 c
14.293 12.387 14.303 9.72 14.302 7.054 c
14.302 6.343 14.354 5.665 15.294 5.648 c
16.061 5.634 16.962 5.377 17.225 6.517 c
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20.218 20.02 20.749 20.442 21.792 20.402 c
22.923 20.359 24.068 20.3 25.189 20.42 c
27.926 20.713 30.241 20.321 31.205 17.271 c
31.242 17.154 31.375 17.069 31.456 16.963 c
33.856 13.78 36.252 10.593 38.656 7.413 c
40.161 5.422 41.478 5.085 43.947 6.055 c
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36.113 17.221 34.735 19.095 33.297 20.92 c
32.492 21.941 32.631 22.71 33.376 23.729 c
36.432 27.908 39.389 32.159 42.397 36.375 c
42.947 37.146 43.56 37.871 44.411 38.961 c
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40.415 39.065 39.778 38.631 39.23 37.875 c
36.234 33.737 33.209 29.618 30.223 25.471 c
29.603 24.61 28.953 24.02 27.785 24.062 c
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19.49 28.125 18.927 30.521 18.389 32.922 c
17.942 34.911 17.474 36.894 17.022 38.852 c
h
95.996 5.618 m
98.506 5.618 l
98.506 30.996 l
98.653 31.041 98.8 31.085 98.947 31.13 c
99.307 30.464 99.721 29.821 100.017 29.128 c
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113.685 5.456 114.213 6.02 114.657 7.12 c
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124.803 5.735 l
128.782 5.735 l
128.782 8.003 l
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121.667 34.867 120.811 32.636 119.996 30.392 c
119.726 30.047 119.367 29.74 119.198 29.351 c
118.106 26.83 117.055 24.292 115.991 21.759 c
115.715 21.101 115.42 20.45 115.175 19.781 c
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112.672 12.915 112.295 12.406 111.992 11.869 c
111.816 11.87 111.64 11.871 111.464 11.872 c
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105.028 26.011 104.1 28.592 103.131 31.157 c
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94.398 5.922 94.848 5.391 95.996 5.618 c
f
Q
0.827 0.514 0.188 rg
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0 0 m
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f
Q
0.043 0.157 0.224 rg
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f
Q
0.82 0.51 0.196 rg
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f
Q
0.827 0.51 0.184 rg
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f
Q
0.824 0.51 0.196 rg
q 1 0 0 1 1412.9441 714.8694 cm
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